Product Data Sheet
Anpirtoline hydrochloride
Catalog No. A45990
Anpirtoline hydrochloride is a selective agonist of the 5-HT1B receptor, exhibiting binding affinities of 28 nM for 5-HT1B, 150 nM for 5-HT1A, and 1.49 μM for 5-HT2 receptors. This compound demonstrates serotonergic activity and displays antinociceptive and antidepressant-like effects. It is valuable for research in neuropharmacology, particularly in studying the role of serotonin receptors in pain modulation and mood disorders.
Chemical Information
| Catalog Num | A45990 |
|---|---|
| M. Wt | 265.21 |
| Formula | C10H14Cl2N2S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 99201-87-3 |
| Synonyms | D-16949 hydrochloride |
| SMILES | ClC1=NC(SC2CCNCC2)=CC=C1.Cl |
Biological Activity
| Description | Anpirtoline hydrochloride is a selective agonist of the 5-HT1B receptor, exhibiting binding affinities of 28 nM for 5-HT1B, 150 nM for 5-HT1A, and 1.49 μM for 5-HT2 receptors. This compound demonstrates serotonergic activity and displays antinociceptive and antidepressant-like effects. It is valuable for research in neuropharmacology, particularly in studying the role of serotonin receptors in pain modulation and mood disorders. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
