Product Data Sheet
Usmarapride free base
Catalog No. A46018
Usmarapride free base is a selective partial agonist of the 5-HT4 receptor, exhibiting a potent activity with an EC50 of 44 nM. This compound is orally active and can penetrate the blood-brain barrier, making it suitable for investigations into cognitive deficits related to Alzheimer's disease. Its mechanism of action supports research aimed at understanding and potentially mitigating Alzheimer's-associated cognitive impairments.
Chemical Information
| Catalog Num | A46018 |
|---|---|
| M. Wt | 383.49 |
| Formula | C21H29N5O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1428862-32-1 |
| Synonyms | SUVN-D4010 free base |
| SMILES | CC(N1N=C(C2=NN=C(C3CCN(CCCOC)CC3)O2)C4=C1C=CC=C4)C |
Biological Activity
| Description | Usmarapride free base is a selective partial agonist of the 5-HT4 receptor, exhibiting a potent activity with an EC50 of 44 nM. This compound is orally active and can penetrate the blood-brain barrier, making it suitable for investigations into cognitive deficits related to Alzheimer's disease. Its mechanism of action supports research aimed at understanding and potentially mitigating Alzheimer's-associated cognitive impairments. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
