Product Data Sheet
Repinotan
Catalog No. A46063
Repinotan is a potent and selective agonist of the 5-HT1A receptor, exhibiting strong brain penetration and oral bioavailability. With Ki values of 0.19 nM in the calf hippocampus, 0.25 nM in rat and human cortex, and 0.59 nM in rat hippocampus, it displays high affinity for target sites while maintaining weak interaction with other related receptors. Repinotan is recognized for its significant neuroprotective properties, making it valuable for research in neuroscience and related therapeutic applications.
Chemical Information
| Catalog Num | A46063 |
|---|---|
| M. Wt | 400.49 |
| Formula | C21H24N2O4S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 144980-29-0 |
| Synonyms | BAY x 3702 free base |
| SMILES | O=C(C1=C2C=CC=C1)N(CCCCNC[C@H]3CCC4=CC=CC=C4O3)S2(=O)=O |
Biological Activity
| Description | Repinotan is a potent and selective agonist of the 5-HT1A receptor, exhibiting strong brain penetration and oral bioavailability. With Ki values of 0.19 nM in the calf hippocampus, 0.25 nM in rat and human cortex, and 0.59 nM in rat hippocampus, it displays high affinity for target sites while maintaining weak interaction with other related receptors. Repinotan is recognized for its significant neuroprotective properties, making it valuable for research in neuroscience and related therapeutic applications. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
