Product Data Sheet
Sumatriptan-d6 succinate
Catalog No. A46089
Sumatriptan-d6 succinate is a deuterated form of Sumatriptan succinate, functioning as an orally active agonist of the 5-HT1 receptor family. With inhibition constants (Kis) of 17 nM, 27 nM, and 100 nM for the 5-HT1D, 5-HT1B, and 5-HT1A receptors, respectively, this compound is primarily utilized in research focused on migraine headaches. Its stable isotope labeling enables advanced studies in pharmacokinetics and metabolism.
Chemical Information
| Catalog Num | A46089 |
|---|---|
| M. Wt | 419.53 |
| Formula | C18H21D6N3O6S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1215621-31-0 |
| Synonyms | GR 43175C-d6 |
| SMILES | OC(CCCC(CC(O)=O)C(O)=O.C(CN(C([2H])([2H])[2H])C([2H])([2H])[2H])C=1C=2C(NC1)=CC=C(CS(NC)(=O)=O)C2 |
Biological Activity
| Description | Sumatriptan-d6 succinate is a deuterated form of Sumatriptan succinate, functioning as an orally active agonist of the 5-HT1 receptor family. With inhibition constants (Kis) of 17 nM, 27 nM, and 100 nM for the 5-HT1D, 5-HT1B, and 5-HT1A receptors, respectively, this compound is primarily utilized in research focused on migraine headaches. Its stable isotope labeling enables advanced studies in pharmacokinetics and metabolism. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
