Product Data Sheet
TC-G 1004
Catalog No. A57909
TC-G 1004 is an orally active antagonist of the A2A adenosine receptor, demonstrating high selectivity with Ki values of 0.44 nM for the human A2A receptor and 80 nM for the human A1 receptor. This compound is valuable in research applications targeting adenosine receptor signaling pathways, particularly in studies related to neurological disorders and cancer. Its efficacy as a selective A2A antagonist makes it a key tool for investigating the role of adenosine receptors in various biological processes.
Chemical Information
| Catalog Num | A57909 |
|---|---|
| M. Wt | 421.50 |
| Formula | C22H27N7O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1061747-72-5 |
| Synonyms | |
| SMILES | CC(NC1=NC(N2N=C(C)C=C2C)=NC(C3=NC(N4CCC(OC)CC4)=CC=C3)=C1)=O |
Biological Activity
| Description | TC-G 1004 is an orally active antagonist of the A2A adenosine receptor, demonstrating high selectivity with Ki values of 0.44 nM for the human A2A receptor and 80 nM for the human A1 receptor. This compound is valuable in research applications targeting adenosine receptor signaling pathways, particularly in studies related to neurological disorders and cancer. Its efficacy as a selective A2A antagonist makes it a key tool for investigating the role of adenosine receptors in various biological processes. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
