Product Data Sheet
A3AR antagonist 4
Catalog No. A57945
A3AR Antagonist 4 is a potent antagonist of the A3 adenosine receptor, exhibiting Ki values of 30.8 nM for the human A3 receptor and 203 nM for the human A1 receptor. This compound is primarily utilized in research focused on cerebral ischemia, enabling investigations into its role in neuroprotection and inflammatory pathways associated with this condition. Through its selective blockade, A3AR Antagonist 4 serves as an important tool for elucidating the therapeutic potential of adenosine receptor modulation in neurological studies.
Chemical Information
| Catalog Num | A57945 |
|---|---|
| M. Wt | 261.28 |
| Formula | C16H11N3O |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 109740-09-2 |
| Synonyms | |
| SMILES | O=C1NC2=C(C=CC=C2)C3=CN(C4=CC=CC=C4)N=C13 |
Biological Activity
| Description | A3AR Antagonist 4 is a potent antagonist of the A3 adenosine receptor, exhibiting Ki values of 30.8 nM for the human A3 receptor and 203 nM for the human A1 receptor. This compound is primarily utilized in research focused on cerebral ischemia, enabling investigations into its role in neuroprotection and inflammatory pathways associated with this condition. Through its selective blockade, A3AR Antagonist 4 serves as an important tool for elucidating the therapeutic potential of adenosine receptor modulation in neurological studies. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
