Product Data Sheet
A2A receptor antagonist 3
Catalog No. A57987
A2A receptor antagonist 3 is a potent adenosine A2A receptor antagonist with a Ki of 0.4 nM. This compound also exhibits binding affinity for A2B, A1, and A3 receptors, with Ki values of 37 nM, 107 nM, and 1467 nM, respectively. It is valuable for research applications involving adenosine signaling pathways and pharmacological studies related to various physiological processes and diseases.
Chemical Information
| Catalog Num | A57987 |
|---|---|
| M. Wt | 454.52 |
| Formula | C26H26N6O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2738606-83-0 |
| Synonyms | |
| SMILES | CC(C)(O)[C@H](C)NC(C1=NC2=C(C3=CC(C)=NC(C)=C3)C(C4=CC(C#N)=CC=C4)=NN2C=C1)=O |
Biological Activity
| Description | A2A receptor antagonist 3 is a potent adenosine A2A receptor antagonist with a Ki of 0.4 nM. This compound also exhibits binding affinity for A2B, A1, and A3 receptors, with Ki values of 37 nM, 107 nM, and 1467 nM, respectively. It is valuable for research applications involving adenosine signaling pathways and pharmacological studies related to various physiological processes and diseases. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
