Product Data Sheet
MRS7799
Catalog No. A58003
MRS7799 is a selective antagonist of the A3 adenosine receptor, demonstrating high affinity with Kds of 0.55 nM for human, 3.74 nM for mouse, and 2.80 nM for rat A3AR. This compound is particularly valuable in research applications related to neurodegeneration, cancer, and ischemic conditions in the heart and brain, as well as autoimmune inflammatory diseases. MRS7799 allows for the exploration of adenosine signaling pathways and their implications in various pathological states.
Chemical Information
| Catalog Num | A58003 |
|---|---|
| M. Wt | 386.47 |
| Formula | C22H18N4OS |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 224040-19-1 |
| Synonyms | DPTN |
| SMILES | O=C(C1=CC=CN=C1)NC2=NC(C3=CC(C)=CC(C)=C3)=C(C4=CC=NC=C4)S2 |
Biological Activity
| Description | MRS7799 is a selective antagonist of the A3 adenosine receptor, demonstrating high affinity with Kds of 0.55 nM for human, 3.74 nM for mouse, and 2.80 nM for rat A3AR. This compound is particularly valuable in research applications related to neurodegeneration, cancer, and ischemic conditions in the heart and brain, as well as autoimmune inflammatory diseases. MRS7799 allows for the exploration of adenosine signaling pathways and their implications in various pathological states. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
