Product Data Sheet
CVT-5440
Catalog No. A58049
CVT-5440 is a selective antagonist of the A2B adenosine receptor, exhibiting high affinity with a Ki value of 50 nM. It demonstrates significant selectivity over other adenosine receptor subtypes, including A1, A2A, and A3, with selectivity ratios greater than 200. This compound is suitable for research applications focusing on asthma and related respiratory conditions, where modulation of adenosine signaling is of interest.
Chemical Information
| Catalog Num | A58049 |
|---|---|
| M. Wt | 516.55 |
| Formula | C27H28N6O5 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 531506-64-6 |
| Synonyms | |
| SMILES | O=C(N1CCC)N(CCC)C2=C(N=C(C3=CC=C(OCC4=NOC(C5=CC=CC(OC)=C5)=N4)C=C3)N2)C1=O |
Biological Activity
| Description | CVT-5440 is a selective antagonist of the A2B adenosine receptor, exhibiting high affinity with a Ki value of 50 nM. It demonstrates significant selectivity over other adenosine receptor subtypes, including A1, A2A, and A3, with selectivity ratios greater than 200. This compound is suitable for research applications focusing on asthma and related respiratory conditions, where modulation of adenosine signaling is of interest. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
