Product Data Sheet
Fipamezole
Catalog No. A58427
Fipamezole is a potent antagonist of the α2-adrenergic receptor, exhibiting Ki values of 9.2 nM, 17 nM, and 55 nM for the human α2A, α2B, and α2C receptors, respectively. This compound serves as an effective anti-dyskinetic agent, making it valuable for research applications in the study of Parkinson's disease and related movement disorders. Its oral bioavailability enhances its utility in various experimental settings.
Chemical Information
| Catalog Num | A58427 |
|---|---|
| M. Wt | 230.28 |
| Formula | C14H15FN2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 150586-58-6 |
| Synonyms | MPV 1730; JP-1730 |
| SMILES | FC1=CC=C2C(CC(C2)(CC)C3=CN=CN3)=C1 |
Biological Activity
| Description | Fipamezole is a potent antagonist of the α2-adrenergic receptor, exhibiting Ki values of 9.2 nM, 17 nM, and 55 nM for the human α2A, α2B, and α2C receptors, respectively. This compound serves as an effective anti-dyskinetic agent, making it valuable for research applications in the study of Parkinson's disease and related movement disorders. Its oral bioavailability enhances its utility in various experimental settings. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
