Product Data Sheet
Azapetine
Catalog No. A58531
Azapetine is an α-adrenergic receptor antagonist that exhibits an IC50 of 0.205 μM for rat α1-adrenergic receptors and 1.3 μM for rat α2-adrenergic receptors. By inhibiting α1 and α2-adrenergic receptor-mediated contractions in blood vessels and vascular smooth muscle, Azapetine serves as a valuable tool for investigating peripheral vascular diseases. Its mechanism of action offers insights into the modulation of vascular tone and potential therapeutic approaches for related disorders.
Chemical Information
| Catalog Num | A58531 |
|---|---|
| M. Wt | 235.32 |
| Formula | C17H17N |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 146-36-1 |
| Synonyms | |
| SMILES | C=CCN1CC2=C(C3=C(C1)C=CC=C3)C=CC=C2 |
Biological Activity
| Description | Azapetine is an α-adrenergic receptor antagonist that exhibits an IC50 of 0.205 μM for rat α1-adrenergic receptors and 1.3 μM for rat α2-adrenergic receptors. By inhibiting α1 and α2-adrenergic receptor-mediated contractions in blood vessels and vascular smooth muscle, Azapetine serves as a valuable tool for investigating peripheral vascular diseases. Its mechanism of action offers insights into the modulation of vascular tone and potential therapeutic approaches for related disorders. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
