Product Data Sheet
Bombesin receptor antagonist-1
Catalog No. A59095
Bombesin receptor antagonist-1 functions as a selective antagonist for the bombesin receptors, exhibiting Ki values of 0.17 nM for the neurotide B (NMB) receptor and 20 nM for the gastrin-releasing peptide (GRP) receptor. This compound is instrumental in the investigation of various pathophysiological conditions, including cancer, depression, and eating disorders. Its precise modulation of bombesin receptors provides valuable insights into receptor signaling pathways and potential therapeutic targets in related diseases.
Chemical Information
| Catalog Num | A59095 |
|---|---|
| M. Wt | 564.68 |
| Formula | C33H36N6O3 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 204067-06-1 |
| Synonyms | |
| SMILES | N#CC(C=C1)=CC=C1NC(N[C@](CC2=CNC3=CC=CC=C23)(C)C(NCC4(C5=CC=C(C=N5)OC)CCCCC4)=O)=O |
Biological Activity
| Description | Bombesin receptor antagonist-1 functions as a selective antagonist for the bombesin receptors, exhibiting Ki values of 0.17 nM for the neurotide B (NMB) receptor and 20 nM for the gastrin-releasing peptide (GRP) receptor. This compound is instrumental in the investigation of various pathophysiological conditions, including cancer, depression, and eating disorders. Its precise modulation of bombesin receptors provides valuable insights into receptor signaling pathways and potential therapeutic targets in related diseases. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
