Product Data Sheet
CB1 antagonist 5
Catalog No. A59364
CB1 Antagonist 5 is a selective antagonist of the cannabinoid receptor type 1 (CB1), exhibiting a Ki value of 243 nM alongside an EC50 of 195 nM. This compound is valuable for research applications targeting the endocannabinoid system and may assist in studies related to pain modulation, appetite regulation, and neuroprotection. Its specificity for the CB1 receptor makes it an essential tool for exploring the physiological roles and therapeutic potentials of cannabinoid signaling.
Chemical Information
| Catalog Num | A59364 |
|---|---|
| M. Wt | 486.16 |
| Formula | C21H14Br2N2O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 878533-35-8 |
| Synonyms | |
| SMILES | O=C1N(C(C(N1C2=CC=C(C=C2)Br)C3=CC=CC=C3)=O)C4=CC=C(C=C4)Br |
Biological Activity
| Description | CB1 Antagonist 5 is a selective antagonist of the cannabinoid receptor type 1 (CB1), exhibiting a Ki value of 243 nM alongside an EC50 of 195 nM. This compound is valuable for research applications targeting the endocannabinoid system and may assist in studies related to pain modulation, appetite regulation, and neuroprotection. Its specificity for the CB1 receptor makes it an essential tool for exploring the physiological roles and therapeutic potentials of cannabinoid signaling. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
