Product Data Sheet
Edonentan hydrate
Catalog No. A60260
Edonentan hydrate is a potent and selective antagonist of the endothelin A (ETA) receptor, exhibiting a high affinity with a Ki value of 10 pM. This compound demonstrates 100% oral bioavailability in rat models, making it an effective tool for in vivo studies. Edonentan hydrate is primarily utilized in research focused on cardiovascular disease and other conditions where endothelin signaling is implicated.
Chemical Information
| Catalog Num | A60260 |
|---|---|
| M. Wt | 554.66 |
| Formula | C28H34N4O6S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 264609-13-4 |
| Synonyms | BMS 207940 hydrate |
| SMILES | CC(C)(C)CC(N(CC1=CC(C2=NC=CO2)=CC=C1C3=CC=CC=C3S(=O)(NC4=NOC(C)=C4C)=O)C)=O.O |
Biological Activity
| Description | Edonentan hydrate is a potent and selective antagonist of the endothelin A (ETA) receptor, exhibiting a high affinity with a Ki value of 10 pM. This compound demonstrates 100% oral bioavailability in rat models, making it an effective tool for in vivo studies. Edonentan hydrate is primarily utilized in research focused on cardiovascular disease and other conditions where endothelin signaling is implicated. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
