Product Data Sheet
Fezagepras
Catalog No. A60330
Fezagepras is a selective modulator of GPR40 and GPR84, functioning as an oral agonist for GPR40 while acting as an antagonist or inverse agonist for GPR84. This compound has demonstrated significant anti-fibrotic, anti-inflammatory, and anti-proliferative activities, effectively reducing renal, liver, and pancreatic fibrosis. Fezagepras holds promise for research related to metabolic disorders and fibrotic diseases, facilitating insights into the roles of GPR40 and GPR84 in various pathological conditions.
Chemical Information
| Catalog Num | A60330 |
|---|---|
| M. Wt | 206.28 |
| Formula | C13H18O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1002101-19-0 |
| Synonyms | Setogepram; PBI-4050 |
| SMILES | O=C(CC1=CC=CC(CCCCC)=C1)O |
Biological Activity
| Description | Fezagepras is a selective modulator of GPR40 and GPR84, functioning as an oral agonist for GPR40 while acting as an antagonist or inverse agonist for GPR84. This compound has demonstrated significant anti-fibrotic, anti-inflammatory, and anti-proliferative activities, effectively reducing renal, liver, and pancreatic fibrosis. Fezagepras holds promise for research related to metabolic disorders and fibrotic diseases, facilitating insights into the roles of GPR40 and GPR84 in various pathological conditions. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
