Product Data Sheet
WAY-207024 dihydrochloride
Catalog No. A60732
WAY-207024 dihydrochloride is a potent antagonist of the gonadotropin-releasing hormone receptor (GnRH-R), exhibiting an IC50 of 12 nM for human GnRH and 71 nM for rat GnRH. This compound effectively inhibits the release of luteinizing hormone (LH) in rats, with an IC50 of 350 nM. WAY-207024 dihydrochloride is useful for studying the regulation of reproductive hormones and exploring therapeutic strategies for disorders related to GnRH signaling.
Chemical Information
| Catalog Num | A60732 |
|---|---|
| M. Wt | 549.54 |
| Formula | C30H34Cl2N6 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 872002-73-8 |
| Synonyms | |
| SMILES | CC(C1=CC=C(C2=NC3=CC=CC(N4CCN(CC5=CC=C6N=CC=NC6=C5)CC4)=C3N2)C=C1)(C)C.[H]Cl.[H]Cl |
Biological Activity
| Description | WAY-207024 dihydrochloride is a potent antagonist of the gonadotropin-releasing hormone receptor (GnRH-R), exhibiting an IC50 of 12 nM for human GnRH and 71 nM for rat GnRH. This compound effectively inhibits the release of luteinizing hormone (LH) in rats, with an IC50 of 350 nM. WAY-207024 dihydrochloride is useful for studying the regulation of reproductive hormones and exploring therapeutic strategies for disorders related to GnRH signaling. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
