Product Data Sheet
GSK256073
Catalog No. A60765
GSK256073 is a potent and selective agonist of the GPR109A receptor, also known as hydroxy-carboxylic acid receptor 2 (HCA2). With a pEC50 of 7.5 in human HCA2, this orally active compound acts as a full agonist without causing flushing. GSK256073 has demonstrated the ability to acutely enhance glucose homeostasis by inhibiting lipolysis, making it a valuable tool for research into type 2 diabetes mellitus (T2DM) and dyslipidemia.
Chemical Information
| Catalog Num | A60765 |
|---|---|
| M. Wt | 256.69 |
| Formula | C10H13ClN4O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 862892-90-8 |
| Synonyms | |
| SMILES | O=C(N(C1=C2NC(Cl)=N1)CCCCC)NC2=O |
Biological Activity
| Description | GSK256073 is a potent and selective agonist of the GPR109A receptor, also known as hydroxy-carboxylic acid receptor 2 (HCA2). With a pEC50 of 7.5 in human HCA2, this orally active compound acts as a full agonist without causing flushing. GSK256073 has demonstrated the ability to acutely enhance glucose homeostasis by inhibiting lipolysis, making it a valuable tool for research into type 2 diabetes mellitus (T2DM) and dyslipidemia. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
