Product Data Sheet
GSK-1292263 hydrochloride
Catalog No. A60791
GSK-1292263 hydrochloride is a potent orally active agonist of GPR119, demonstrating a pEC50 of approximately 6.9 nM for human GPR119 and 6.7 nM for rat GPR119. This compound is primarily utilized in research focused on type 2 diabetes and dyslipidemia, contributing to a better understanding of metabolic regulation and potential therapeutic interventions. Its ability to activate GPR119 makes it a valuable tool for exploring signaling pathways and metabolic processes influenced by this receptor.
Chemical Information
| Catalog Num | A60791 |
|---|---|
| M. Wt | 493.02 |
| Formula | C23H29ClN4O4S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1032824-54-6 |
| Synonyms | |
| SMILES | CC(C1=NOC(N2CCC(CC2)COC3=CN=C(C=C3)C4=CC=C(C=C4)S(C)(=O)=O)=N1)C.[H]Cl |
Biological Activity
| Description | GSK-1292263 hydrochloride is a potent orally active agonist of GPR119, demonstrating a pEC50 of approximately 6.9 nM for human GPR119 and 6.7 nM for rat GPR119. This compound is primarily utilized in research focused on type 2 diabetes and dyslipidemia, contributing to a better understanding of metabolic regulation and potential therapeutic interventions. Its ability to activate GPR119 makes it a valuable tool for exploring signaling pathways and metabolic processes influenced by this receptor. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
