Product Data Sheet
GPR139 agonist-2
Catalog No. A60797
GPR139 agonist-2 is a selective agonist targeting the GPR139 receptor, demonstrating a potent EC50 of 24.7 nM. This compound has shown promising biological activity by rescuing social interaction deficits and ameliorating cognitive impairments in murine models of schizophrenia. GPR139 agonist-2 holds potential for use in antipsychotic drug research and the exploration of novel therapeutic strategies for schizophrenia.
Chemical Information
| Catalog Num | A60797 |
|---|---|
| M. Wt | 380.32 |
| Formula | C17H15F3N4O3 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2983118-29-0 |
| Synonyms | |
| SMILES | O=C1N(CC(N[C@@H](C)C2=CC=C(OC(F)(F)F)C=C2)=O)N=CC3=CC=CN31 |
Biological Activity
| Description | GPR139 agonist-2 is a selective agonist targeting the GPR139 receptor, demonstrating a potent EC50 of 24.7 nM. This compound has shown promising biological activity by rescuing social interaction deficits and ameliorating cognitive impairments in murine models of schizophrenia. GPR139 agonist-2 holds potential for use in antipsychotic drug research and the exploration of novel therapeutic strategies for schizophrenia. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
