GPR81 agonist 2
Catalog No. A60906

GPR81 Agonist 2 specifically targets the GPR81 receptor, exhibiting potent agonistic activity with EC50 values of 0.023 µM for human GPR81 and 0.123 µM for human GPR109A. This compound is valuable for research in metabolic regulation, insulin sensitivity, and tumor metabolism. Its ability to selectively activate GPR81 makes it a useful tool for probing signaling pathways related to energy homeostasis and lipid metabolism.
Chemical Information
| Catalog Num | A60906 |
|---|---|
| M. Wt | 603.11 |
| Formula | C26H27ClN6O5S2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1143024-28-5 |
| Synonyms | |
| SMILES | O=C(NC1=NC2=C(S1)C=C(S(=O)(C3CCN(CC3)C)=O)C=C2)NC(C4=C(Cl)C=C(OCC)C(N5N=CC=C5)=C4)=O |
Biological Activity
| Description | GPR81 Agonist 2 specifically targets the GPR81 receptor, exhibiting potent agonistic activity with EC50 values of 0.023 µM for human GPR81 and 0.123 µM for human GPR109A. This compound is valuable for research in metabolic regulation, insulin sensitivity, and tumor metabolism. Its ability to selectively activate GPR81 makes it a useful tool for probing signaling pathways related to energy homeostasis and lipid metabolism. |
|---|
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Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.


