Product Data Sheet
CP-96021
Catalog No. A60996
CP-96021 is a potent antagonist of the leukotriene D4 (LTD4) receptor (Ki = 34 μM) and the platelet activating factor (PAF) receptor (Ki = 37 μM). This compound effectively targets two key inflammatory mediators, making it valuable in research on inflammation-related pathologies. With a high specificity profile, CP-96021 demonstrates negligible activity against various receptors, including dopamine, adenosine, and GABA receptors, suggesting minimal off-target effects. This reagent can be employed in studies investigating the pathogenesis of inflammatory diseases, such as asthma.
Chemical Information
| Catalog Num | A60996 |
|---|---|
| M. Wt | 492.57 |
| Formula | C29H21FN4OS |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 139401-43-7 |
| Synonyms | |
| SMILES | CC1=NC2=CN=CC=C2N1C3=CC=C(C=C3)OCC4=CC(/C=C/C5=NC6=CC(F)=CC=C6S5)=CC=C4 |
Biological Activity
| Description | CP-96021 is a potent antagonist of the leukotriene D4 (LTD4) receptor (Ki = 34 μM) and the platelet activating factor (PAF) receptor (Ki = 37 μM). This compound effectively targets two key inflammatory mediators, making it valuable in research on inflammation-related pathologies. With a high specificity profile, CP-96021 demonstrates negligible activity against various receptors, including dopamine, adenosine, and GABA receptors, suggesting minimal off-target effects. This reagent can be employed in studies investigating the pathogenesis of inflammatory diseases, such as asthma. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
