Product Data Sheet
hMC1R agonist 1
Catalog No. A61662
hMC1R Agonist 1 selectively activates the human melanocortin 1 receptor (hMC1R) with an EC50 of 3 nM. This compound demonstrates over 300-fold selectivity for hMC1R compared to hMC3R, hMC4R, and hMC5R, which have significantly higher EC50 values (902 nM, 915 nM, and >1000 nM, respectively). hMC1R Agonist 1 holds promise for potential therapeutic applications within the melanocortin receptor family, particularly in conditions related to pigmentation and metabolic regulation.
Chemical Information
| Catalog Num | A61662 |
|---|---|
| M. Wt | 1107.35 |
| Formula | C54H70N14O8S2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 3028881-87-7 |
| Synonyms | |
| SMILES |
Biological Activity
| Description | hMC1R Agonist 1 selectively activates the human melanocortin 1 receptor (hMC1R) with an EC50 of 3 nM. This compound demonstrates over 300-fold selectivity for hMC1R compared to hMC3R, hMC4R, and hMC5R, which have significantly higher EC50 values (902 nM, 915 nM, and >1000 nM, respectively). hMC1R Agonist 1 holds promise for potential therapeutic applications within the melanocortin receptor family, particularly in conditions related to pigmentation and metabolic regulation. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
