Product Data Sheet
MPCI
Catalog No. A61713
MPCI is a selective antagonist of the melanocortin-4 receptor (MC4R), exhibiting pharmacological chaperone activity. With a Ki value of 0.218 μM determined in HEK293 cells expressing human MC4R, MPCI is valuable in researching the mechanisms underlying MC4R-deficient obesity. This compound can facilitate studies on metabolic regulation and potential therapeutic approaches for related disorders.
Chemical Information
| Catalog Num | A61713 |
|---|---|
| M. Wt | 519.45 |
| Formula | C25H32BrFN4O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 884538-31-2 |
| Synonyms | |
| SMILES | O=C(C1=CC=CC(F)=C1CCC2=CC(Br)=CC=C2OC)NC(NCC3CCN(CC3)CC)=N |
Biological Activity
| Description | MPCI is a selective antagonist of the melanocortin-4 receptor (MC4R), exhibiting pharmacological chaperone activity. With a Ki value of 0.218 μM determined in HEK293 cells expressing human MC4R, MPCI is valuable in researching the mechanisms underlying MC4R-deficient obesity. This compound can facilitate studies on metabolic regulation and potential therapeutic approaches for related disorders. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
