Product Data Sheet
GR 87389
Catalog No. A62115
GR 87389 is a potent antagonist of the NK2 receptor, effectively inhibiting its activity. This compound has been shown to competitively block GA 64349-induced contractions in smooth muscle strips derived from human detrusor, prostate, and prostatic urethra tissues. GR 87389 is valuable in research applications focused on the role of NK2 receptors in smooth muscle physiology and potential therapeutic strategies for related disorders.
Chemical Information
| Catalog Num | A62115 |
|---|---|
| M. Wt | 900.07 |
| Formula | C47H65N9O9 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 141663-86-7 |
| Synonyms | |
| SMILES | CCCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H]1CCCN1C(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)OC(C)(C)C)C(N)=O |
Biological Activity
| Description | GR 87389 is a potent antagonist of the NK2 receptor, effectively inhibiting its activity. This compound has been shown to competitively block GA 64349-induced contractions in smooth muscle strips derived from human detrusor, prostate, and prostatic urethra tissues. GR 87389 is valuable in research applications focused on the role of NK2 receptors in smooth muscle physiology and potential therapeutic strategies for related disorders. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
