M617
Catalog No. A62193

M617 is a selective galanin receptor 1 (GAL1) agonist, exhibiting inhibition constants (Kis) of 0.23 nM and 5.71 nM for GAL1 and GAL2, respectively. This compound primarily targets GAL1 to promote GLUT4 expression, significantly enhancing GLUT4 content in the cardiac muscle of type 2 diabetic rats. M617 is useful in research focused on metabolic disorders and the modulation of glucose homeostasis.
Chemical Information
| Catalog Num | A62193 |
|---|---|
| M. Wt | 2361.65 |
| Formula | C112H161N29O28 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 860790-38-1 |
| Synonyms | |
| SMILES | C([C@@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(NCC(N[C@@H](CC1=CC=C(O)C=C1)C(N[C@H](C(N[C@H](C(NCC(=O)N2[C@H](C(N[C@H](C(=O)N3[C@H](C(=O)N4[C@H](C(NCC(N[C@@H](CC5=CC=CC=C5)C(N[C@H](C(=O)N6[C@H](C(N[C@@H](CC7=CC=CC=C7)C(N[C@@H](CCCNC(=N)N)C(N)=O)=O)=O)CCC6)CO)=O)=O)=O)CCC4)CCC3)CCC(N)=O)=O)CCC2)=O)CC(C)C)=O)CC(C)C)=O)=O)=O)C)=O)CO)=O)CC(N)=O)=O)CC(C)C)=O)[C@@H](C)O)=O)NC(CN)=O)C=8C=9C(NC8)=CC=CC9 |
Biological Activity
| Description | M617 is a selective galanin receptor 1 (GAL1) agonist, exhibiting inhibition constants (Kis) of 0.23 nM and 5.71 nM for GAL1 and GAL2, respectively. This compound primarily targets GAL1 to promote GLUT4 expression, significantly enhancing GLUT4 content in the cardiac muscle of type 2 diabetic rats. M617 is useful in research focused on metabolic disorders and the modulation of glucose homeostasis. |
|---|
RETURN POLICY
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Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.


