Spiradoline mesylate
Catalog No. A62363

Spiradoline mesylate is a selective kappa-opioid receptor (KOR) agonist with a Ki of 8.6 nM, demonstrating strong receptor affinity. It exhibits significant diuretic, analgesic, antiarrhythmic, antitussive, and neuroprotective activities, allowing it to effectively penetrate the blood-brain barrier. This compound is valuable for research applications focusing on pain management, addiction studies, and neuroprotection related to opioid activity.
Chemical Information
| Catalog Num | A62363 |
|---|---|
| M. Wt | 521.50 |
| Formula | C23H34Cl2N2O5S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 87173-97-5 |
| Synonyms | U-62066 mesylate |
| SMILES | ClC1=C(C=CC(CC(N([C@H]2CC[C@@]3(C[C@@H]2N4CCCC4)OCCC3)C)=O)=C1)Cl.CS(O)(=O)=O |
Biological Activity
| Description | Spiradoline mesylate is a selective kappa-opioid receptor (KOR) agonist with a Ki of 8.6 nM, demonstrating strong receptor affinity. It exhibits significant diuretic, analgesic, antiarrhythmic, antitussive, and neuroprotective activities, allowing it to effectively penetrate the blood-brain barrier. This compound is valuable for research applications focusing on pain management, addiction studies, and neuroprotection related to opioid activity. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.


