Product Data Sheet
EST73502 monohydrochloride
Catalog No. A62396
EST73502 monohydrochloride acts as a selective μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, exhibiting Kis of 64 nM and 118 nM for each target, respectively. This compound is orally bioavailable and can effectively cross the blood-brain barrier. EST73502 demonstrates notable antinociceptive properties, making it a valuable tool for research into pain modulation and neurobiology.
Chemical Information
| Catalog Num | A62396 |
|---|---|
| M. Wt | 388.88 |
| Formula | C19H27ClF2N2O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2535970-65-9 |
| Synonyms | |
| SMILES | FC1=CC=C(F)C=C1CCN(CC2)CCC2(O[C@@H]3C)CN(CC)C3=O.[H]Cl |
Biological Activity
| Description | EST73502 monohydrochloride acts as a selective μ-opioid receptor (MOR) agonist and σ1 receptor (σ1R) antagonist, exhibiting Kis of 64 nM and 118 nM for each target, respectively. This compound is orally bioavailable and can effectively cross the blood-brain barrier. EST73502 demonstrates notable antinociceptive properties, making it a valuable tool for research into pain modulation and neurobiology. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
