Product Data Sheet
Picenadol
Catalog No. A62460
Picenadol is an opioid mixed agonist-antagonist that primarily targets the μ-opioid receptor. The compound consists of a racemic mixture, with the d-isomer functioning as a potent μ-opioid receptor agonist and the l-isomer acting as a weak competitive antagonist, which diminishes the agonist effect and mitigates the risk of dependence. Additionally, Picenadol exhibits anticholinergic activity, making it relevant for research applications in pain management and opioid pharmacology.
Chemical Information
| Catalog Num | A62460 |
|---|---|
| M. Wt | 247.38 |
| Formula | C16H25NO |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 79201-85-7 |
| Synonyms | LY-150720 |
| SMILES | CCC[C@]1([C@@H](C)CN(CC1)C)C2=CC(O)=CC=C2 |
Biological Activity
| Description | Picenadol is an opioid mixed agonist-antagonist that primarily targets the μ-opioid receptor. The compound consists of a racemic mixture, with the d-isomer functioning as a potent μ-opioid receptor agonist and the l-isomer acting as a weak competitive antagonist, which diminishes the agonist effect and mitigates the risk of dependence. Additionally, Picenadol exhibits anticholinergic activity, making it relevant for research applications in pain management and opioid pharmacology. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
