Product Data Sheet
CR 665 acetate
Catalog No. A62497
CR 665 acetate is a selective kappa-opioid receptor agonist that targets opioid receptors to effectively manage visceral pain. By activating receptors on afferent nerves within the gut, CR 665 acetate enhances pain tolerance without the central nervous system effects typical of non-selective opioids. This compound is particularly useful in the context of postoperative pain management, offering a fast-acting analgesic alternative without the delayed response associated with other opioids. Its peripheral selectivity may provide significant advantages in pain relief while minimizing potential side effects.
Chemical Information
| Catalog Num | A62497 |
|---|---|
| M. Wt | 731.88 |
| Formula | C38H53N9O6 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 958873-83-1 |
| Synonyms | JNJ 38488502 acetate; FE 200665 acetate |
| SMILES | N=C(N)NCCC[C@H](C(N)=O)N(C([C@@H](CCCC)NC([C@@H](CC1=CC=CC=C1)NC([C@@H](CC2=CC=CC=C2)N)=O)=O)=O)CC3=CC=NC=C3.CC(O)=O |
Biological Activity
| Description | CR 665 acetate is a selective kappa-opioid receptor agonist that targets opioid receptors to effectively manage visceral pain. By activating receptors on afferent nerves within the gut, CR 665 acetate enhances pain tolerance without the central nervous system effects typical of non-selective opioids. This compound is particularly useful in the context of postoperative pain management, offering a fast-acting analgesic alternative without the delayed response associated with other opioids. Its peripheral selectivity may provide significant advantages in pain relief while minimizing potential side effects. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
