Product Data Sheet
BPRMU191
Catalog No. A62526
BPRMU191 is a selective μ-opioid receptor (MOR) modulator that transforms small-molecule morphinan antagonists into G protein-biased MOR agonists. This conversion facilitates MOR-dependent activation, resulting in potent analgesic effects while minimizing adverse side effects such as gastrointestinal issues, antinociceptive tolerance, and dependency risks. BPRMU191, when used in conjunction with morphinan antagonists, provides a valuable tool for exploring severe pain management and the modulation of G protein-coupled receptors in research settings.
Chemical Information
| Catalog Num | A62526 |
|---|---|
| M. Wt | 331.36 |
| Formula | C17H14FNO3S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2131199-52-3 |
| Synonyms | |
| SMILES | O=C(C1=CC=C(N2C(CSC2C3=CC=C(C=C3)F)=O)C(C)=C1)O |
Biological Activity
| Description | BPRMU191 is a selective μ-opioid receptor (MOR) modulator that transforms small-molecule morphinan antagonists into G protein-biased MOR agonists. This conversion facilitates MOR-dependent activation, resulting in potent analgesic effects while minimizing adverse side effects such as gastrointestinal issues, antinociceptive tolerance, and dependency risks. BPRMU191, when used in conjunction with morphinan antagonists, provides a valuable tool for exploring severe pain management and the modulation of G protein-coupled receptors in research settings. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
