Product Data Sheet
Mu opioid receptor antagonist 2
Catalog No. A62528
Mu Opioid Receptor Antagonist 2 is a highly potent and selective antagonist of the μ opioid receptor (MOR), exhibiting a Ki of 0.37 nM and an EC50 of 0.44 nM. This compound effectively penetrates the blood-brain barrier and demonstrates strong central nervous system antagonism against morphine, inducing fewer withdrawal symptoms compared to traditional remedies. Mu Opioid Receptor Antagonist 2 is valuable for research focused on opioid use disorders (OUD), enabling a better understanding of opioid dependency and potential therapeutic interventions.
Chemical Information
| Catalog Num | A62528 |
|---|---|
| M. Wt | 452.57 |
| Formula | C25H28N2O4S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2773925-64-5 |
| Synonyms | |
| SMILES | O[C@]12[C@H]3CC4=C5[C@@]1(CCN3CC6CC6)[C@H]([C@H](CC2)NC(C7=CC=CS7)=O)OC5=C(O)C=C4 |
Biological Activity
| Description | Mu Opioid Receptor Antagonist 2 is a highly potent and selective antagonist of the μ opioid receptor (MOR), exhibiting a Ki of 0.37 nM and an EC50 of 0.44 nM. This compound effectively penetrates the blood-brain barrier and demonstrates strong central nervous system antagonism against morphine, inducing fewer withdrawal symptoms compared to traditional remedies. Mu Opioid Receptor Antagonist 2 is valuable for research focused on opioid use disorders (OUD), enabling a better understanding of opioid dependency and potential therapeutic interventions. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
