Product Data Sheet
Mu opioid receptor antagonist 7
Catalog No. A62562
Mu opioid receptor antagonist 7 is a potent antagonist of the µ-opioid receptor (µOR), demonstrating an IC50 value of 29 ± 3.0 nM. This compound is highly permeable to the central nervous system, making it suitable for investigating pain mechanisms and the pharmacology of opioid use disorder. Its efficacy in modulating µOR activity supports its use in preclinical research settings focused on opioid receptor signaling and related therapeutic interventions.
Chemical Information
| Catalog Num | A62562 |
|---|---|
| M. Wt | 386.91 |
| Formula | C22H27ClN2O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2378397-30-7 |
| Synonyms | |
| SMILES | OC1=CC(Cl)=C(C[C@H](N(C)C)CNC([C@@H]2C[C@]2(C)C3=CC=CC=C3)=O)C=C1 |
Biological Activity
| Description | Mu opioid receptor antagonist 7 is a potent antagonist of the µ-opioid receptor (µOR), demonstrating an IC50 value of 29 ± 3.0 nM. This compound is highly permeable to the central nervous system, making it suitable for investigating pain mechanisms and the pharmacology of opioid use disorder. Its efficacy in modulating µOR activity supports its use in preclinical research settings focused on opioid receptor signaling and related therapeutic interventions. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
