Product Data Sheet
DBPR116
Catalog No. A62583
DBPR116 is a prodrug of BPRMU191 designed for efficient penetration of the blood-brain barrier. This compound enhances the delivery of centrally acting analgesics and has been shown to provide superior safety and analgesic efficacy in combination with Naltrexone compared to traditional opioids such as morphine. In various in vivo pharmacological models, DBPR116 effectively alleviates pain related to thermal and cancer sources while minimizing adverse effects, suggesting its potential as a safer alternative in opioid analgesia.
Chemical Information
| Catalog Num | A62583 |
|---|---|
| M. Wt | 359.41 |
| Formula | C19H18FNO3S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2131200-75-2 |
| Synonyms | |
| SMILES | O=C(C1=CC=C(N2C(CSC2C3=CC=C(C=C3)F)=O)C(C)=C1)OCC |
Biological Activity
| Description | DBPR116 is a prodrug of BPRMU191 designed for efficient penetration of the blood-brain barrier. This compound enhances the delivery of centrally acting analgesics and has been shown to provide superior safety and analgesic efficacy in combination with Naltrexone compared to traditional opioids such as morphine. In various in vivo pharmacological models, DBPR116 effectively alleviates pain related to thermal and cancer sources while minimizing adverse effects, suggesting its potential as a safer alternative in opioid analgesia. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
