Product Data Sheet
MOR agonist-5
Catalog No. A62630
MOR agonist-5 is a selective and potent mu-opioid receptor (MOR) agonist, exhibiting an EC50 of 0.25 nM. It demonstrates a significantly lower affinity for delta-opioid receptors (DOR) with an EC50 of 10 nM, and a negligible effect on kappa-opioid receptors (KOR) and nociceptin/orphanin FQ peptide receptors (NOR) at concentrations exceeding 10,000 nM. MOR agonist-5 displays substantial antinociceptive properties, making it a valuable tool for research into pain management and opioid receptor pharmacology.
Chemical Information
| Catalog Num | A62630 |
|---|---|
| M. Wt | 349.47 |
| Formula | C22H27N3O |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 3085132-31-3 |
| Synonyms | |
| SMILES | NC(C1=CC(N2[C@H]3CC[C@@H]2CN(CCCC4=CC=CC=C4)C3)=CC=C1)=O |
Biological Activity
| Description | MOR agonist-5 is a selective and potent mu-opioid receptor (MOR) agonist, exhibiting an EC50 of 0.25 nM. It demonstrates a significantly lower affinity for delta-opioid receptors (DOR) with an EC50 of 10 nM, and a negligible effect on kappa-opioid receptors (KOR) and nociceptin/orphanin FQ peptide receptors (NOR) at concentrations exceeding 10,000 nM. MOR agonist-5 displays substantial antinociceptive properties, making it a valuable tool for research into pain management and opioid receptor pharmacology. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
