Product Data Sheet
L-367773
Catalog No. A62765
L-367773 is a selective antagonist of the oxytocin receptor, demonstrating Ki values of 26 nM for the rat uterine oxytocin receptor and 61 nM for the human uterine oxytocin receptor. This compound effectively inhibits oxytocin-stimulated uterine contractions, making it a valuable tool for research related to reproductive biology and uterine physiology. Its oral bioactivity further enhances its utility in pharmacological studies.
Chemical Information
| Catalog Num | A62765 |
|---|---|
| M. Wt | 510.69 |
| Formula | C28H38N4O3S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 152140-41-5 |
| Synonyms | |
| SMILES | O=C(N[C@@H]1[C@](C2(C)C)(CS(=O)(N3CCC4(CC3)CCC5=C4C=CC=C5)=O)CC[C@]2([H])C1)CC6=CNC=N6 |
Biological Activity
| Description | L-367773 is a selective antagonist of the oxytocin receptor, demonstrating Ki values of 26 nM for the rat uterine oxytocin receptor and 61 nM for the human uterine oxytocin receptor. This compound effectively inhibits oxytocin-stimulated uterine contractions, making it a valuable tool for research related to reproductive biology and uterine physiology. Its oral bioactivity further enhances its utility in pharmacological studies. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
