Product Data Sheet
EP3 antagonist 2
Catalog No. A63375
EP3 antagonist 2 is a potent and selective antagonist of the EP3 receptor, exhibiting a strong binding affinity with a Ki value of 3.3 nM. This compound demonstrates significant antagonistic activity, with an IC50 of 30.8 nM, as determined by its ability to modulate cellular cAMP levels. EP3 antagonist 2 is suitable for research applications exploring the physiological roles of the EP3 receptor in various biological processes and potential therapeutic interventions.
Chemical Information
| Catalog Num | A63375 |
|---|---|
| M. Wt | 347.41 |
| Formula | C21H21N3O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1952261-87-8 |
| Synonyms | |
| SMILES | O=C1C([C@]2(C)C(NCCC2)=O)=CC=C(C3=CC4=C(C)C=CC=C4N=C3)N1 |
Biological Activity
| Description | EP3 antagonist 2 is a potent and selective antagonist of the EP3 receptor, exhibiting a strong binding affinity with a Ki value of 3.3 nM. This compound demonstrates significant antagonistic activity, with an IC50 of 30.8 nM, as determined by its ability to modulate cellular cAMP levels. EP3 antagonist 2 is suitable for research applications exploring the physiological roles of the EP3 receptor in various biological processes and potential therapeutic interventions. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
