Product Data Sheet
PAR-2 antagonist 1
Catalog No. A63490
PAR-2 antagonist 1 is a selective antagonist of protease-activated receptor 2 (PAR2), exhibiting an inhibitory concentration IC50 value of 0.9 μM. This compound effectively blocks PAR2 signaling, which is implicated in the proliferation and migration of breast cancer cells. PAR-2 antagonist 1 is valuable for research applications focused on understanding PAR2's role in cancer biology and exploring potential therapeutic strategies for breast cancer treatment.
Chemical Information
| Catalog Num | A63490 |
|---|---|
| M. Wt | 406.48 |
| Formula | C27H22N2O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 3119609-65-0 |
| Synonyms | |
| SMILES | O=C(N/C(C(NCC1=CC=CC=C1)=O)=C\C2=CC=CC3=C2C=CC=C3)C4=CC=CC=C4 |
Biological Activity
| Description | PAR-2 antagonist 1 is a selective antagonist of protease-activated receptor 2 (PAR2), exhibiting an inhibitory concentration IC50 value of 0.9 μM. This compound effectively blocks PAR2 signaling, which is implicated in the proliferation and migration of breast cancer cells. PAR-2 antagonist 1 is valuable for research applications focused on understanding PAR2's role in cancer biology and exploring potential therapeutic strategies for breast cancer treatment. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
