Product Data Sheet
BN-81674
Catalog No. A63881
BN-81674 is a selective antagonist targeting the human somatostatin sst3 receptor, exhibiting a Ki of 0.92 nM. This compound effectively reverses the inhibition of cyclic AMP accumulation caused by somatostatin at nanomolar concentrations, with an IC50 value of 0.84 nM. BN-81674 is suitable for applications in cancer research, particularly in studies assessing somatostatin signaling pathways and their implications in tumor biology.
Chemical Information
| Catalog Num | A63881 |
|---|---|
| M. Wt | 454.65 |
| Formula | C30H38N4 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 252278-73-2 |
| Synonyms | |
| SMILES | CCCCCC1(N[C@H](CC2=C1NC3=C2C=CC=C3)C4=NC=C(N4)C5=CC=CC=C5)CCCCC |
Biological Activity
| Description | BN-81674 is a selective antagonist targeting the human somatostatin sst3 receptor, exhibiting a Ki of 0.92 nM. This compound effectively reverses the inhibition of cyclic AMP accumulation caused by somatostatin at nanomolar concentrations, with an IC50 value of 0.84 nM. BN-81674 is suitable for applications in cancer research, particularly in studies assessing somatostatin signaling pathways and their implications in tumor biology. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
