Product Data Sheet
PK-THPP
Catalog No. A68004
PK-THPP is a selective blocker of the TASK-3 potassium ion channel (K2P9.1), exhibiting IC50 values of 35 nM for TASK-3 and 300 nM for TASK-1. This compound demonstrates minimal activity against other potassium channels, making it a valuable tool for investigating specific ion channel functions. PK-THPP is recognized for its efficacy as a breathing stimulant and is useful for research into various breathing disorders and related physiological studies.
Chemical Information
| Catalog Num | A68004 |
|---|---|
| M. Wt | 468.59 |
| Formula | C29H32N4O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1332454-07-5 |
| Synonyms | |
| SMILES | O=C(C1=CC=C(C2=CC=CC=C2)C=C1)N3CC4=C(N5CCC(C(CCC)=O)CC5)N=CN=C4CC3 |
Biological Activity
| Description | PK-THPP is a selective blocker of the TASK-3 potassium ion channel (K2P9.1), exhibiting IC50 values of 35 nM for TASK-3 and 300 nM for TASK-1. This compound demonstrates minimal activity against other potassium channels, making it a valuable tool for investigating specific ion channel functions. PK-THPP is recognized for its efficacy as a breathing stimulant and is useful for research into various breathing disorders and related physiological studies. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
