Product Data Sheet
TRPV1 antagonist 3
Catalog No. A68727
TRPV1 antagonist 3 (Compound 7q) is a highly effective antagonist of the TRPV1 receptor, demonstrating an IC50 of 2.66 nM against capsaicin. This compound exhibits mode-selectivity and is characterized by favorable oral bioavailability (F = 60%) as well as the ability to penetrate the central nervous system. TRPV1 antagonist 3 is valuable for research focused on pain modulation and inflammatory processes.
Chemical Information
| Catalog Num | A68727 |
|---|---|
| M. Wt | 391.53 |
| Formula | C23H25N3OS |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2765294-54-8 |
| Synonyms | |
| SMILES | CC(C1=CC=CC(NC(N2CCC[C@H]2C3=NC=C(S3)C4=CC=CC=C4)=O)=C1)C |
Biological Activity
| Description | TRPV1 antagonist 3 (Compound 7q) is a highly effective antagonist of the TRPV1 receptor, demonstrating an IC50 of 2.66 nM against capsaicin. This compound exhibits mode-selectivity and is characterized by favorable oral bioavailability (F = 60%) as well as the ability to penetrate the central nervous system. TRPV1 antagonist 3 is valuable for research focused on pain modulation and inflammatory processes. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
