Product Data Sheet
LEI-101 free base
Catalog No. A73392
LEI-101 free base is a selective and orally bioavailable agonist of the CB2 receptor, primarily targeting inflammation and oxidative stress-related conditions. It demonstrates a binding potency to CB2 receptors that is approximately 100 times greater than its affinity for CB1 receptors, with a pEC50 value of 8. The compound’s pharmacological profile suggests potential applications in the treatment of diseases such as kidney disease, making it valuable in therapeutic research.
Chemical Information
| Catalog Num | A73392 |
|---|---|
| M. Wt | 472.53 |
| Formula | C23H25FN4O4S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 1228660-00-1 |
| Synonyms | |
| SMILES | O=C1N(C(CN1CC2=CC=C(C=C2)C3=NC(CN(CC4)CCS4(=O)=O)=C(C=C3)F)=O)C5CC5 |
Biological Activity
| Description | LEI-101 free base is a selective and orally bioavailable agonist of the CB2 receptor, primarily targeting inflammation and oxidative stress-related conditions. It demonstrates a binding potency to CB2 receptors that is approximately 100 times greater than its affinity for CB1 receptors, with a pEC50 value of 8. The compound’s pharmacological profile suggests potential applications in the treatment of diseases such as kidney disease, making it valuable in therapeutic research. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
