Product Data Sheet

EST64454

Catalog No. A79292

main product photo
EST64454 is a selective sigma-1 receptor antagonist with a Ki value of 22 nM, demonstrating oral bioactivity. This compound is useful for investigating pain mechanisms and signaling pathways associated with sigma-1 receptor activity. Its application in research can provide insights into pain modulation and potential therapeutic interventions.
Chemical Information
Catalog NumA79292
M. Wt364.39
FormulaC18H22F2N4O2
Purity>98%
Storageat -20 °C 3 years (powder form); at -20 °C 6 months (Solution base)
CAS No.1351438-26-0
Synonyms
SMILESCC(N1CCN(CCOCC2=NN(C3=CC=C(F)C(F)=C3)C=C2)CC1)=O
Biological Activity
DescriptionEST64454 is a selective sigma-1 receptor antagonist with a Ki value of 22 nM, demonstrating oral bioactivity. This compound is useful for investigating pain mechanisms and signaling pathways associated with sigma-1 receptor activity. Its application in research can provide insights into pain modulation and potential therapeutic interventions.
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SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.