Product Data Sheet
UniPR500
Catalog No. A84705
UniPR500 is a competitive antagonist of the EphA2 receptor, exhibiting a Ki value of 0.78 μM. This compound effectively inhibits the binding of biotinylated ephrin-A1 to EphA2 in a dose-dependent manner, with an IC50 of 1.1 μM. UniPR500 is valuable for research applications focusing on cellular signaling pathways and the role of EphA2 in various diseases.
Chemical Information
| Catalog Num | A84705 |
|---|---|
| M. Wt | 589.81 |
| Formula | C36H51N3O4 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2085767-98-0 |
| Synonyms | |
| SMILES | C[C@@]12[C@](CC[C@]2([H])[C@H](C)CCC(N[C@H](CC(O)=O)CC3=CNC4=CC=CC=C34)=O)([H])[C@@]5([H])[C@@](CC1)([H])[C@@]6([C@](C/C(CC6)=N/O)([H])CC5)C |
Biological Activity
| Description | UniPR500 is a competitive antagonist of the EphA2 receptor, exhibiting a Ki value of 0.78 μM. This compound effectively inhibits the binding of biotinylated ephrin-A1 to EphA2 in a dose-dependent manner, with an IC50 of 1.1 μM. UniPR500 is valuable for research applications focusing on cellular signaling pathways and the role of EphA2 in various diseases. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
