Product Data Sheet
KSL 128114
Catalog No. A84821
KSL 128114 is a potent peptide inhibitor of syntenin, targeting the PDZ1 domain with nanomolar affinity. This compound exhibits stability in human plasma and mouse hepatic microsomes, making it suitable for in vitro and in vivo studies. KSL 128114 demonstrates selective inhibition of syntenin, providing valuable insights into cellular signaling pathways and potential therapeutic applications in disorders associated with syntenin dysregulation.
Chemical Information
| Catalog Num | A84821 |
|---|---|
| M. Wt | 2201.59 |
| Formula | C96H165N39O21 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2757292-12-7 |
| Synonyms | |
| SMILES | C([C@H](NC([C@H](CC1=CN=CN1)NC([C@@H](NC([C@H](NC([C@@H](NC([C@H](NC([C@@H](NC([C@H](NC(CNC([C@H](NC([C@@H](NC([C@@H](CCCNC(=N)N)NC(C)=O)=O)CCCNC(=N)N)=O)CCCNC(=N)N)=O)=O)CCCNC(=N)N)=O)CCCCN)=O)CCCCN)=O)CCCNC(=N)N)=O)CCCNC(=N)N)=O)CO)=O)=O)C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@@H]([C@H](CC)C)C(O)=O)=O)CC(O)=O)=O)C2CCCCC2)=O)[C@](C)(C)C)=O)C=3C=4C(NC3)=CC=CC4 |
Biological Activity
| Description | KSL 128114 is a potent peptide inhibitor of syntenin, targeting the PDZ1 domain with nanomolar affinity. This compound exhibits stability in human plasma and mouse hepatic microsomes, making it suitable for in vitro and in vivo studies. KSL 128114 demonstrates selective inhibition of syntenin, providing valuable insights into cellular signaling pathways and potential therapeutic applications in disorders associated with syntenin dysregulation. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
