Product Data Sheet
EPI-7170
Catalog No. A84925
EPI-7170 is a potent androgen receptor (AR) antagonist that targets the N-terminal structural domain of the receptor. It effectively inhibits the transcriptional activity of full-length androgen receptor (FL-AR) and its splice variants, providing therapeutic potential against enzalutamide-resistant castration-resistant prostate cancer (CRPC). This compound is valuable for research into mechanisms of resistance in prostate cancer and the development of novel therapeutic strategies.
Chemical Information
| Catalog Num | A84925 |
|---|---|
| M. Wt | 540.88 |
| Formula | C22H28Cl3NO6S |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2139288-26-7 |
| Synonyms | |
| SMILES | CC(C1=CC(Cl)=C(C(Cl)=C1)OC[C@H](O)CCl)(C2=CC=C(C=C2)OC[C@H](O)CNS(C)(=O)=O)C |
Biological Activity
| Description | EPI-7170 is a potent androgen receptor (AR) antagonist that targets the N-terminal structural domain of the receptor. It effectively inhibits the transcriptional activity of full-length androgen receptor (FL-AR) and its splice variants, providing therapeutic potential against enzalutamide-resistant castration-resistant prostate cancer (CRPC). This compound is valuable for research into mechanisms of resistance in prostate cancer and the development of novel therapeutic strategies. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
