Product Data Sheet
AR antagonist 5
Catalog No. A85024
AR Antagonist 5 is a selective antagonist of the androgen receptor, exhibiting an IC50 value of 134.8 nM. This compound demonstrates favorable pharmacokinetic properties, characterized by high skin exposure and low plasma exposure. AR Antagonist 5 is valuable for research applications targeting androgen receptor signaling pathways in various biological studies related to hormone regulation and therapeutic interventions in androgen-sensitive conditions.
Chemical Information
| Catalog Num | A85024 |
|---|---|
| M. Wt | 470.45 |
| Formula | C23H21F3N6O2 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2902679-53-0 |
| Synonyms | |
| SMILES | C[C@](CN1CC2CC(N2C3=CC=C(C=C3)C#N)C1)(C(NC4=CN=C(C(C(F)(F)F)=C4)C#N)=O)O |
Biological Activity
| Description | AR Antagonist 5 is a selective antagonist of the androgen receptor, exhibiting an IC50 value of 134.8 nM. This compound demonstrates favorable pharmacokinetic properties, characterized by high skin exposure and low plasma exposure. AR Antagonist 5 is valuable for research applications targeting androgen receptor signaling pathways in various biological studies related to hormone regulation and therapeutic interventions in androgen-sensitive conditions. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
