Product Data Sheet
Taragarestrant meglumine
Catalog No. A85109
Taragarestrant meglumine is a selective estrogen receptor degrader (SERD) known for its potent activity against estrogen receptors. This compound effectively inhibits the growth of estrogen receptor-positive (ER+) breast cancer cell lines and demonstrates significant efficacy in xenograft models. It serves as a valuable tool for research into targeted therapies for ER+ breast cancer, aiding in the understanding of estrogen receptor biology and the potential for innovative treatment strategies.
Chemical Information
| Catalog Num | A85109 |
|---|---|
| M. Wt | 670.60 |
| Formula | C32H42Cl2FN3O7 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 2446618-18-2 |
| Synonyms | D-0502 meglumine |
| SMILES | CC(C)(F)CN1[C@@](C2=C(C=C(C=C2Cl)/C=C/C(O)=O)Cl)([H])C3=C(C[C@H]1C)C4=CC=CC=C4N3.OC[C@@H](O)[C@@H](O)[C@H](O)[C@@H](O)CNC |
Biological Activity
| Description | Taragarestrant meglumine is a selective estrogen receptor degrader (SERD) known for its potent activity against estrogen receptors. This compound effectively inhibits the growth of estrogen receptor-positive (ER+) breast cancer cell lines and demonstrates significant efficacy in xenograft models. It serves as a valuable tool for research into targeted therapies for ER+ breast cancer, aiding in the understanding of estrogen receptor biology and the potential for innovative treatment strategies. |
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RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
