Product Data Sheet

Androgen receptor allosteric antagonist 1

Catalog No. A85179

main product photo
Androgen Receptor Allosteric Antagonist 1 is a competitive allosteric inhibitor of the androgen receptor, exhibiting a Ki of 9 μM. This compound effectively inhibits R1881-mediated transcriptional activity and cell proliferation, making it a valuable tool for studying prostate cancer. Its unique mechanism of action allows for detailed exploration of androgen receptor signaling pathways in cancer research.
Chemical Information
Catalog NumA85179
M. Wt336.43
FormulaC21H24N2O2
Purity>98%
Storageat -20 °C 3 years (powder form); at -20 °C 6 months (Solution base)
CAS No.927819-39-4
Synonyms
SMILESO=C(CC1=CN(CC(C)C)C2=CC=C(C3=C(OC)C=CC=C3)C=C21)N
Biological Activity
DescriptionAndrogen Receptor Allosteric Antagonist 1 is a competitive allosteric inhibitor of the androgen receptor, exhibiting a Ki of 9 μM. This compound effectively inhibits R1881-mediated transcriptional activity and cell proliferation, making it a valuable tool for studying prostate cancer. Its unique mechanism of action allows for detailed exploration of androgen receptor signaling pathways in cancer research.
RETURN POLICY
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SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.