Product Data Sheet
CMP8
Catalog No. A85239
CMP8 is a selective ligand for the estrogen receptor, specifically targeting the mutant estrogen receptor ligand binding domain (ERLBD). This compound demonstrates potent biological activity with IC50 values of 29 nM for MGERα, 41 nM for MGRERα, 1100 nM for human ERα, and 2200 nM for human ERβ. CMP8 is valuable for research applications focused on estrogen receptor modulation and its role in cancer biology.
Chemical Information
| Catalog Num | A85239 |
|---|---|
| M. Wt | 528.08 |
| Formula | C33H34ClNO3 |
| Purity | >98% |
| Storage | at -20 °C 3 years (powder form); at -20 °C 6 months (Solution base) |
| CAS No. | 851107-28-3 |
| Synonyms | |
| SMILES | O=C1CCC2(CC3=CC=C(Cl)C=C3)CC4=C(C=CC(O)=C4)C2=C1C5=CC=C(OCCN6CCCCC6)C=C5 |
Biological Activity
| Description | CMP8 is a selective ligand for the estrogen receptor, specifically targeting the mutant estrogen receptor ligand binding domain (ERLBD). This compound demonstrates potent biological activity with IC50 values of 29 nM for MGERα, 41 nM for MGRERα, 1100 nM for human ERα, and 2200 nM for human ERβ. CMP8 is valuable for research applications focused on estrogen receptor modulation and its role in cancer biology. |
|---|
RETURN POLICY
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
Adooq’s Unconditional Return Policy ensures a smooth online shopping experience for our customers. If you are in any way unsatisfied with your purchase, you may return any item(s) within 7 days of receiving it. In the event of product quality issues, either protocol related or product related problems, you may return any item(s) within 365 days from the original purchase date. Please follow the instructions below when returning products.
SHIPPING AND STORAGE
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
Adooq products are transported at room temperature. If you receive the product at room temperature, please rest assured, the Adooq Quality Inspection Department has conducted experiments to verify that the normal temperature placement of one month will not affect the biological activity of powder products. After collecting, please store the product according to the requirements described in the datasheet. Most Adooq products are stable under the recommended conditions.
