Apatinib (YN968D1)

Apatinib (YN968D1) is a tyrosine kinase inhibitor that selectively inhibits the vascular endothelial growth factor receptor-2 (VEGFR2, also known as KDR) that inhibits VEGF-mediated endothelial cell migration and proliferation thus blocking new blood vessel formation in tumor tissue.
Grouped product items
Product Name Price Stock Qty
Apatinib 5mg
$100.00
In stock
Apatinib 10mg
$150.00
In stock
Apatinib 50mg
$350.00
In stock
Apatinib 100mg
$450.00
In stock
Apatinib (YN968D1) 10mM * 1mL in DMSO
$110.00
In stock
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Adooq Products cited in reputable paper
Adooq's Apatinib (YN968D1) has been cited by 2 publications
  • Wonjin Park, .et al. , Biomed Pharmacother, 2021, Feb;134:111110 PMID: 33338749
  • Majid Momeny, .et al. , Sci Rep, 2017, 7: 45954 PMID: 28383032
  • Biological Activity
    Discription Apatinib (YN968D1) is a tyrosine kinase inhibitor that selectively inhibits the vascular endothelial growth factor receptor-2 (VEGFR2, also known as KDR) that inhibits VEGF-mediated endothelial cell migration and proliferation thus blocking new blood vessel formation in tumor tissue.
    Targets
    Target Value
    Product Information
    Catalog Num A11407
    Formula C25H27N5O4S
    Molecular Weight 493.6
    CAS Number 811803-05-1
    SMILES CS(=O)(=O)O.C1CCC(C1)(C#N)C2=CC=C(C=C2)NC(=O)C3=C(N=CC=C3)NCC4=CC=NC=C4
    Storage

    Store lyophilized at -20ºC, keep desiccated.
    In lyophilized form, the chemical is stable for 36 months.
    In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

    Solubility
    In vitro DMSO 77 mg/mL (193.72 mM)
    Water Insoluble
    Ethanol 10 mg/mL
    * <1 mg/ml means slightly soluble or insoluble.
    * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
    Preparing Stock Solutions
    Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
    0.1 mM 20.26 mL 101.3 mL 202.59 mL
    0.5 mM 4.05 mL 20.26 mL 40.52 mL
    1 mM 2.03 mL 10.13 mL 20.26 mL
    5 mM 0.41 mL 2.03 mL 4.05 mL
    Useful Calculator

    This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

    Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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    Please check COA/MSDS for correct molecular weight.

    Calculate the dilution required to prepare a stock solution.
    This equation is commonly abbreviated as: C1V1 = C2V2

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